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INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology
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Zeitschriftentitel: | ACS Medicinal Chemistry Letters |
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Personen und Körperschaften: | , , , , , , , , , , , , , , , , , , , , , , , , , |
In: | ACS Medicinal Chemistry Letters, 8, 2017, 5, S. 486-491 |
Format: | E-Article |
Sprache: | Englisch |
veröffentlicht: |
American Chemical Society (ACS)
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Schlagwörter: |
author_facet |
Yue, Eddy W. Sparks, Richard Polam, Padmaja Modi, Dilip Douty, Brent Wayland, Brian Glass, Brian Takvorian, Amy Glenn, Joseph Zhu, Wenyu Bower, Michael Liu, Xiangdong Leffet, Lynn Wang, Qian Bowman, Kevin J. Hansbury, Michael J. Wei, Min Li, Yanlong Wynn, Richard Burn, Timothy C. Koblish, Holly K. Fridman, Jordan S. Emm, Tom Scherle, Peggy A. Metcalf, Brian Combs, Andrew P. Yue, Eddy W. Sparks, Richard Polam, Padmaja Modi, Dilip Douty, Brent Wayland, Brian Glass, Brian Takvorian, Amy Glenn, Joseph Zhu, Wenyu Bower, Michael Liu, Xiangdong Leffet, Lynn Wang, Qian Bowman, Kevin J. Hansbury, Michael J. Wei, Min Li, Yanlong Wynn, Richard Burn, Timothy C. Koblish, Holly K. Fridman, Jordan S. Emm, Tom Scherle, Peggy A. Metcalf, Brian Combs, Andrew P. |
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author |
Yue, Eddy W. Sparks, Richard Polam, Padmaja Modi, Dilip Douty, Brent Wayland, Brian Glass, Brian Takvorian, Amy Glenn, Joseph Zhu, Wenyu Bower, Michael Liu, Xiangdong Leffet, Lynn Wang, Qian Bowman, Kevin J. Hansbury, Michael J. Wei, Min Li, Yanlong Wynn, Richard Burn, Timothy C. Koblish, Holly K. Fridman, Jordan S. Emm, Tom Scherle, Peggy A. Metcalf, Brian Combs, Andrew P. |
spellingShingle |
Yue, Eddy W. Sparks, Richard Polam, Padmaja Modi, Dilip Douty, Brent Wayland, Brian Glass, Brian Takvorian, Amy Glenn, Joseph Zhu, Wenyu Bower, Michael Liu, Xiangdong Leffet, Lynn Wang, Qian Bowman, Kevin J. Hansbury, Michael J. Wei, Min Li, Yanlong Wynn, Richard Burn, Timothy C. Koblish, Holly K. Fridman, Jordan S. Emm, Tom Scherle, Peggy A. Metcalf, Brian Combs, Andrew P. ACS Medicinal Chemistry Letters INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology Organic Chemistry Drug Discovery Biochemistry |
author_sort |
yue, eddy w. |
spelling |
Yue, Eddy W. Sparks, Richard Polam, Padmaja Modi, Dilip Douty, Brent Wayland, Brian Glass, Brian Takvorian, Amy Glenn, Joseph Zhu, Wenyu Bower, Michael Liu, Xiangdong Leffet, Lynn Wang, Qian Bowman, Kevin J. Hansbury, Michael J. Wei, Min Li, Yanlong Wynn, Richard Burn, Timothy C. Koblish, Holly K. Fridman, Jordan S. Emm, Tom Scherle, Peggy A. Metcalf, Brian Combs, Andrew P. 1948-5875 1948-5875 American Chemical Society (ACS) Organic Chemistry Drug Discovery Biochemistry http://dx.doi.org/10.1021/acsmedchemlett.6b00391 INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology ACS Medicinal Chemistry Letters |
doi_str_mv |
10.1021/acsmedchemlett.6b00391 |
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American Chemical Society (ACS) |
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title |
INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology |
title_unstemmed |
INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology |
title_full |
INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology |
title_fullStr |
INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology |
title_full_unstemmed |
INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology |
title_short |
INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology |
title_sort |
incb24360 (epacadostat), a highly potent and selective indoleamine-2,3-dioxygenase 1 (ido1) inhibitor for immuno-oncology |
topic |
Organic Chemistry Drug Discovery Biochemistry |
url |
http://dx.doi.org/10.1021/acsmedchemlett.6b00391 |
publishDate |
2017 |
physical |
486-491 |
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author | Yue, Eddy W., Sparks, Richard, Polam, Padmaja, Modi, Dilip, Douty, Brent, Wayland, Brian, Glass, Brian, Takvorian, Amy, Glenn, Joseph, Zhu, Wenyu, Bower, Michael, Liu, Xiangdong, Leffet, Lynn, Wang, Qian, Bowman, Kevin J., Hansbury, Michael J., Wei, Min, Li, Yanlong, Wynn, Richard, Burn, Timothy C., Koblish, Holly K., Fridman, Jordan S., Emm, Tom, Scherle, Peggy A., Metcalf, Brian, Combs, Andrew P. |
author_facet | Yue, Eddy W., Sparks, Richard, Polam, Padmaja, Modi, Dilip, Douty, Brent, Wayland, Brian, Glass, Brian, Takvorian, Amy, Glenn, Joseph, Zhu, Wenyu, Bower, Michael, Liu, Xiangdong, Leffet, Lynn, Wang, Qian, Bowman, Kevin J., Hansbury, Michael J., Wei, Min, Li, Yanlong, Wynn, Richard, Burn, Timothy C., Koblish, Holly K., Fridman, Jordan S., Emm, Tom, Scherle, Peggy A., Metcalf, Brian, Combs, Andrew P., Yue, Eddy W., Sparks, Richard, Polam, Padmaja, Modi, Dilip, Douty, Brent, Wayland, Brian, Glass, Brian, Takvorian, Amy, Glenn, Joseph, Zhu, Wenyu, Bower, Michael, Liu, Xiangdong, Leffet, Lynn, Wang, Qian, Bowman, Kevin J., Hansbury, Michael J., Wei, Min, Li, Yanlong, Wynn, Richard, Burn, Timothy C., Koblish, Holly K., Fridman, Jordan S., Emm, Tom, Scherle, Peggy A., Metcalf, Brian, Combs, Andrew P. |
author_sort | yue, eddy w. |
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publisher | American Chemical Society (ACS) |
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spelling | Yue, Eddy W. Sparks, Richard Polam, Padmaja Modi, Dilip Douty, Brent Wayland, Brian Glass, Brian Takvorian, Amy Glenn, Joseph Zhu, Wenyu Bower, Michael Liu, Xiangdong Leffet, Lynn Wang, Qian Bowman, Kevin J. Hansbury, Michael J. Wei, Min Li, Yanlong Wynn, Richard Burn, Timothy C. Koblish, Holly K. Fridman, Jordan S. Emm, Tom Scherle, Peggy A. Metcalf, Brian Combs, Andrew P. 1948-5875 1948-5875 American Chemical Society (ACS) Organic Chemistry Drug Discovery Biochemistry http://dx.doi.org/10.1021/acsmedchemlett.6b00391 INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology ACS Medicinal Chemistry Letters |
spellingShingle | Yue, Eddy W., Sparks, Richard, Polam, Padmaja, Modi, Dilip, Douty, Brent, Wayland, Brian, Glass, Brian, Takvorian, Amy, Glenn, Joseph, Zhu, Wenyu, Bower, Michael, Liu, Xiangdong, Leffet, Lynn, Wang, Qian, Bowman, Kevin J., Hansbury, Michael J., Wei, Min, Li, Yanlong, Wynn, Richard, Burn, Timothy C., Koblish, Holly K., Fridman, Jordan S., Emm, Tom, Scherle, Peggy A., Metcalf, Brian, Combs, Andrew P., ACS Medicinal Chemistry Letters, INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology, Organic Chemistry, Drug Discovery, Biochemistry |
title | INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology |
title_full | INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology |
title_fullStr | INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology |
title_full_unstemmed | INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology |
title_short | INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology |
title_sort | incb24360 (epacadostat), a highly potent and selective indoleamine-2,3-dioxygenase 1 (ido1) inhibitor for immuno-oncology |
title_unstemmed | INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology |
topic | Organic Chemistry, Drug Discovery, Biochemistry |
url | http://dx.doi.org/10.1021/acsmedchemlett.6b00391 |